4e47
SET7/9 in complex with inhibitor (R)-(3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6- sulfonamide and S-adenosylmethionineSET7/9 in complex with inhibitor (R)-(3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6- sulfonamide and S-adenosylmethionine
Structural highlights
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OCACategories:
- Histone-lysine N-methyltransferase
- Homo sapiens
- Arrowsmith, C H.
- Barsyte, D.
- Bountra, C.
- Brown, P J.
- Bunnage, M.
- Cook, A.
- Dong, A.
- Edwards, A M.
- Fish, P.
- Ouyang, H.
- Owen, D.
- SGC, Structural Genomics Consortium.
- Tatlock, J.
- Vedadi, M.
- Walker, J R.
- Weigelt, J.
- Chromatin regulator
- Chromosomal protein
- Inhibitor
- Methyltransferase
- Nucleus
- S-adenosylmethionine
- Set domain
- Sgc
- Structural genomics consortium
- Ternary complex
- Transcription
- Transcription regulation
- Transferase
- Transferase-transferase inhibitor complex