2r7b: Difference between revisions
New page: '''Unreleased structure''' The entry 2r7b is ON HOLD until Sep 07 2009 Authors: Olland, A.M. Description: Crystal Structure of the Phosphoinositide-dependent Kinase-1 (PDK-1)Catalytic ... |
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===Crystal Structure of the Phosphoinositide-dependent Kinase-1 (PDK-1)Catalytic Domain bound to a dibenzonaphthyridine inhibitor=== | |||
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''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Wed | ==About this Structure== | ||
2R7B is a [[Single protein]] structure of sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=2R7B OCA]. | |||
==Reference== | |||
Discovery of dibenzo[c,f][2,7]naphthyridines as potent and selective 3-phosphoinositide-dependent kinase-1 inhibitors., Gopalsamy A, Shi M, Boschelli DH, Williamson R, Olland A, Hu Y, Krishnamurthy G, Han X, Arndt K, Guo B, J Med Chem. 2007 Nov 15;50(23):5547-9. Epub 2007 Oct 17. PMID:[http://www.ncbi.nlm.nih.gov/pubmed/17941624 17941624] | |||
[[Category: Homo sapiens]] | |||
[[Category: Non-specific serine/threonine protein kinase]] | |||
[[Category: Single protein]] | |||
[[Category: Olland, A M.]] | |||
[[Category: Dibenzonaphthyridine]] | |||
[[Category: Inhibitor]] | |||
[[Category: Pdk1]] | |||
[[Category: Signaling protein]] | |||
[[Category: Structure]] | |||
[[Category: Transferase]] | |||
''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Wed Sep 10 10:41:37 2008'' |