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| [[Image:2vin.jpg|left|200px]] | | [[Image:2vin.jpg|left|200px]] |
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| {{Structure
| | <!-- |
| |PDB= 2vin |SIZE=350|CAPTION= <scene name='initialview01'>2vin</scene>, resolution 1.9Å
| | The line below this paragraph, containing "STRUCTURE_2vin", creates the "Structure Box" on the page. |
| |SITE= <scene name='pdbsite=AC1:Act+Binding+Site+For+Chain+A'>AC1</scene>, <scene name='pdbsite=AC2:So4+Binding+Site+For+Chain+A'>AC2</scene> and <scene name='pdbsite=AC3:505+Binding+Site+For+Chain+A'>AC3</scene>
| | You may change the PDB parameter (which sets the PDB file loaded into the applet) |
| |LIGAND= <scene name='pdbligand=505:(2R)-1-(2,6-DIMETHYLPHENOXY)PROPAN-2-AMINE'>505</scene>, <scene name='pdbligand=ACT:ACETATE+ION'>ACT</scene>, <scene name='pdbligand=SO4:SULFATE+ION'>SO4</scene>
| | or the SCENE parameter (which sets the initial scene displayed when the page is loaded), |
| |ACTIVITY= <span class='plainlinks'>[http://en.wikipedia.org/wiki/U-plasminogen_activator U-plasminogen activator], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=3.4.21.73 3.4.21.73] </span>
| | or leave the SCENE parameter empty for the default display. |
| |GENE= | | --> |
| |DOMAIN= | | {{STRUCTURE_2vin| PDB=2vin | SCENE= }} |
| |RELATEDENTRY=[[1c5w|1C5W]], [[1c5x|1C5X]], [[1c5y|1C5Y]], [[1c5z|1C5Z]], [[1ejn|1EJN]], [[1fv9|1FV9]], [[1gi7|1GI7]], [[1gi9|1GI9]], [[1gj7|1GJ7]], [[1gj8|1GJ8]], [[1gj9|1GJ9]], [[1gjc|1GJC]], [[1kdu|1KDU]], [[1o5c|1O5C]], [[1owd|1OWD]], [[1owh|1OWH]], [[1owj|1OWJ]], [[1sc8|1SC8]], [[1f5l|1F5L]], [[1f92|1F92]], [[1gi8|1GI8]], [[1gja|1GJA]], [[1gjb|1GJB]], [[1gjd|1GJD]], [[1lmw|1LMW]], [[1o3p|1O3P]], [[1o5a|1O5A]], [[1o5b|1O5B]], [[1owe|1OWE]], [[1owi|1OWI]], [[1owk|1OWK]], [[1sqa|1SQA]], [[1sqo|1SQO]], [[1sqt|1SQT]], [[1u6q|1U6Q]], [[1vj9|1VJ9]], [[1w0z|1W0Z]], [[1w10|1W10]], [[1w12|1W12]], [[1w14|1W14]], [[1vja|1VJA]], [[1w11|1W11]], [[1w13|1W13]], [[2jde|2JDE]], [[2vio|2VIO]], [[2vip|2VIP]], [[2viq|2VIQ]], [[2viv|2VIV]], [[2viw|2VIW]]
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| |RESOURCES=<span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=2vin FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=2vin OCA], [http://www.ebi.ac.uk/pdbsum/2vin PDBsum], [http://www.rcsb.org/pdb/explore.do?structureId=2vin RCSB]</span>
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| }} | |
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| '''FRAGMENT-BASED DISCOVERY OF MEXILETINE DERIVATIVES AS ORALLY BIOAVAILABLE INHIBITORS OF UROKINASE-TYPE PLASMINOGEN ACTIVATOR''' | | '''FRAGMENT-BASED DISCOVERY OF MEXILETINE DERIVATIVES AS ORALLY BIOAVAILABLE INHIBITORS OF UROKINASE-TYPE PLASMINOGEN ACTIVATOR''' |
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| [[Category: Vinkovic, M.]] | | [[Category: Vinkovic, M.]] |
| [[Category: Wallis, N G.]] | | [[Category: Wallis, N G.]] |
| [[Category: blood coagulation]] | | [[Category: Blood coagulation]] |
| [[Category: egf-like domain]] | | [[Category: Egf-like domain]] |
| [[Category: fibrinolysis]] | | [[Category: Fibrinolysis]] |
| [[Category: glycoprotein]] | | [[Category: Glycoprotein]] |
| [[Category: hydrolase]] | | [[Category: Hydrolase]] |
| [[Category: inhibitor]] | | [[Category: Inhibitor]] |
| [[Category: kringle]] | | [[Category: Kringle]] |
| [[Category: pharmaceutical]] | | [[Category: Pharmaceutical]] |
| [[Category: phosphorylation]] | | [[Category: Phosphorylation]] |
| [[Category: plasminogen activation]] | | [[Category: Plasminogen activation]] |
| [[Category: polymorphism]] | | [[Category: Polymorphism]] |
| [[Category: protease]] | | [[Category: Protease]] |
| [[Category: secreted]] | | [[Category: Secreted]] |
| [[Category: serine protease]] | | [[Category: Serine protease]] |
| [[Category: urokinase-type plasminogen activator]] | | [[Category: Urokinase-type plasminogen activator]] |
| [[Category: zymogen]] | | [[Category: Zymogen]] |
| | | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Sun May 4 18:52:47 2008'' |
| ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Mon Mar 31 05:12:47 2008'' | |