1vyw: Difference between revisions

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|PDB= 1vyw |SIZE=350|CAPTION= <scene name='initialview01'>1vyw</scene>, resolution 2.30&Aring;
|PDB= 1vyw |SIZE=350|CAPTION= <scene name='initialview01'>1vyw</scene>, resolution 2.30&Aring;
|SITE= <scene name='pdbsite=DG1:So4+Binding+Site+For+Chain+D'>DG1</scene>
|SITE= <scene name='pdbsite=DG1:So4+Binding+Site+For+Chain+D'>DG1</scene>
|LIGAND= <scene name='pdbligand=SO4:SULFATE+ION'>SO4</scene> and <scene name='pdbligand=292:N-(3-CYCLOPROPYL-1H-PYRAZOL-5-YL)-2-(2-NAPHTHYL)ACETAMIDE'>292</scene>
|LIGAND= <scene name='pdbligand=292:N-(3-CYCLOPROPYL-1H-PYRAZOL-5-YL)-2-(2-NAPHTHYL)ACETAMIDE'>292</scene>, <scene name='pdbligand=SO4:SULFATE+ION'>SO4</scene>
|ACTIVITY= [http://en.wikipedia.org/wiki/Transferred_entry:_2.7.11.1 Transferred entry: 2.7.11.1], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.1.37 2.7.1.37]  
|ACTIVITY= <span class='plainlinks'>[http://en.wikipedia.org/wiki/Non-specific_serine/threonine_protein_kinase Non-specific serine/threonine protein kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.11.1 2.7.11.1] </span>
|GENE=  
|GENE=  
|DOMAIN=
|RELATEDENTRY=
|RESOURCES=<span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=1vyw FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=1vyw OCA], [http://www.ebi.ac.uk/pdbsum/1vyw PDBsum], [http://www.rcsb.org/pdb/explore.do?structureId=1vyw RCSB]</span>
}}
}}


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3-Aminopyrazole inhibitors of CDK2/cyclin A as antitumor agents. 1. Lead finding., Pevarello P, Brasca MG, Amici R, Orsini P, Traquandi G, Corti L, Piutti C, Sansonna P, Villa M, Pierce BS, Pulici M, Giordano P, Martina K, Fritzen EL, Nugent RA, Casale E, Cameron A, Ciomei M, Roletto F, Isacchi A, Fogliatto G, Pesenti E, Pastori W, Marsiglio A, Leach KL, Clare PM, Fiorentini F, Varasi M, Vulpetti A, Warpehoski MA, J Med Chem. 2004 Jun 17;47(13):3367-80. PMID:[http://www.ncbi.nlm.nih.gov/pubmed/15189033 15189033]
3-Aminopyrazole inhibitors of CDK2/cyclin A as antitumor agents. 1. Lead finding., Pevarello P, Brasca MG, Amici R, Orsini P, Traquandi G, Corti L, Piutti C, Sansonna P, Villa M, Pierce BS, Pulici M, Giordano P, Martina K, Fritzen EL, Nugent RA, Casale E, Cameron A, Ciomei M, Roletto F, Isacchi A, Fogliatto G, Pesenti E, Pastori W, Marsiglio A, Leach KL, Clare PM, Fiorentini F, Varasi M, Vulpetti A, Warpehoski MA, J Med Chem. 2004 Jun 17;47(13):3367-80. PMID:[http://www.ncbi.nlm.nih.gov/pubmed/15189033 15189033]
[[Category: Homo sapiens]]
[[Category: Homo sapiens]]
[[Category: Non-specific serine/threonine protein kinase]]
[[Category: Protein complex]]
[[Category: Protein complex]]
[[Category: Transferred entry: 2 7.11 1]]
[[Category: Amici, R.]]
[[Category: Amici, R.]]
[[Category: Brasca, M G.]]
[[Category: Brasca, M G.]]
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[[Category: Vulpetti, A.]]
[[Category: Vulpetti, A.]]
[[Category: Warpehoski, M A.]]
[[Category: Warpehoski, M A.]]
[[Category: 292]]
[[Category: SO4]]
[[Category: cell division]]
[[Category: cell division]]
[[Category: cyclin]]
[[Category: cyclin]]
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[[Category: transferase]]
[[Category: transferase]]


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