4pp7: Difference between revisions
No edit summary |
No edit summary |
||
Line 1: | Line 1: | ||
==Highly Potent and Selective 3-N-methylquinazoline-4(3H)-one Based Inhibitors of B-RafV600E Kinase== | ==Highly Potent and Selective 3-N-methylquinazoline-4(3H)-one Based Inhibitors of B-RafV600E Kinase== | ||
<StructureSection load='4pp7' size='340' side='right' caption='[[4pp7]], [[Resolution|resolution]] 3.40Å' scene=''> | <StructureSection load='4pp7' size='340' side='right' caption='[[4pp7]], [[Resolution|resolution]] 3.40Å' scene=''> | ||
Line 6: | Line 7: | ||
<tr id='gene'><td class="sblockLbl"><b>[[Gene|Gene:]]</b></td><td class="sblockDat">BRAF, BRAF1, RAFB1 ([http://www.ncbi.nlm.nih.gov/Taxonomy/Browser/wwwtax.cgi?mode=Info&srchmode=5&id=9606 HUMAN])</td></tr> | <tr id='gene'><td class="sblockLbl"><b>[[Gene|Gene:]]</b></td><td class="sblockDat">BRAF, BRAF1, RAFB1 ([http://www.ncbi.nlm.nih.gov/Taxonomy/Browser/wwwtax.cgi?mode=Info&srchmode=5&id=9606 HUMAN])</td></tr> | ||
<tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Non-specific_serine/threonine_protein_kinase Non-specific serine/threonine protein kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.11.1 2.7.11.1] </span></td></tr> | <tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Non-specific_serine/threonine_protein_kinase Non-specific serine/threonine protein kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.11.1 2.7.11.1] </span></td></tr> | ||
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4pp7 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=4pp7 OCA], [http://www.rcsb.org/pdb/explore.do?structureId=4pp7 RCSB], [http://www.ebi.ac.uk/pdbsum/4pp7 PDBsum]</span></td></tr> | <tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4pp7 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=4pp7 OCA], [http://pdbe.org/4pp7 PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=4pp7 RCSB], [http://www.ebi.ac.uk/pdbsum/4pp7 PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=4pp7 ProSAT]</span></td></tr> | ||
</table> | </table> | ||
== Disease == | == Disease == | ||
Line 20: | Line 21: | ||
From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine.<br> | From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine.<br> | ||
</div> | </div> | ||
<div class="pdbe-citations 4pp7" style="background-color:#fffaf0;"></div> | |||
==See Also== | ==See Also== |