3rpy: Difference between revisions
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==CDK2 in complex with inhibitor RC-2-40== | ==CDK2 in complex with inhibitor RC-2-40== | ||
<StructureSection load='3rpy' size='340' side='right' caption='[[3rpy]], [[Resolution|resolution]] 1.90Å' scene=''> | <StructureSection load='3rpy' size='340' side='right' caption='[[3rpy]], [[Resolution|resolution]] 1.90Å' scene=''> | ||
== Structural highlights == | == Structural highlights == | ||
<table><tr><td colspan='2'>[[3rpy]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/ | <table><tr><td colspan='2'>[[3rpy]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Human Human]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=3RPY OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=3RPY FirstGlance]. <br> | ||
</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=27Z:4-AMINO-2-[(4-SULFAMOYLPHENYL)AMINO]-1,3-THIAZOLE-5-CARBOXAMIDE'>27Z</scene></td></tr> | </td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=27Z:4-AMINO-2-[(4-SULFAMOYLPHENYL)AMINO]-1,3-THIAZOLE-5-CARBOXAMIDE'>27Z</scene></td></tr> | ||
<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[3ql8|3ql8]], [[3qqf|3qqf]], [[3qqg|3qqg]], [[3qqh|3qqh]], [[3qqj|3qqj]], [[3qqk|3qqk]], [[3qql|3qql]], [[3qrt|3qrt]], [[3qru|3qru]], [[3qtq|3qtq]], [[3qtr|3qtr]], [[3qts|3qts]], [[3qtu|3qtu]], [[3qtw|3qtw]], [[3qtx|3qtx]], [[3qtz|3qtz]], [[3qu0|3qu0]], [[3qwj|3qwj]], [[3qwk|3qwk]], [[3qx2|3qx2]], [[3qx4|3qx4]], [[3qxo|3qxo]], [[3qxp|3qxp]], [[3qzf|3qzf]], [[3qzg|3qzg]], [[3qzh|3qzh]], [[3qzi|3qzi]], [[3r1q|3r1q]], [[3r1s|3r1s]], [[3r1y|3r1y]], [[3r28|3r28]], [[3r6x|3r6x]], [[3r71|3r71]], [[3r73|3r73]], [[3r7e|3r7e]], [[3r7i|3r7i]], [[3r7u|3r7u]], [[3r7v|3r7v]], [[3r7y|3r7y]], [[3r83|3r83]], [[3r8l|3r8l]], [[3r8m|3r8m]], [[3r8p|3r8p]], [[3r8u|3r8u]], [[3r8v|3r8v]], [[3r8z|3r8z]], [[3r9d|3r9d]], [[3r9h|3r9h]], [[3r9n|3r9n]], [[3r9o|3r9o]], [[3rah|3rah]], [[3rai|3rai]], [[3rak|3rak]], [[3ral|3ral]], [[3rjc|3rjc]], [[3rk5|3rk5]], [[3rk7|3rk7]], [[3rk9|3rk9]], [[3rkb|3rkb]], [[3rm6|3rm6]], [[3rm7|3rm7]], [[3rmf|3rmf]], [[3rni|3rni]], [[3roy|3roy]], [[3rpo|3rpo]], [[3rpr|3rpr]], [[3rpv|3rpv]], [[3rzb|3rzb]], [[3s00|3s00]], [[3s0o|3s0o]], [[3s1h|3s1h]], [[3sqq|3sqq]]</td></tr> | <tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[3ql8|3ql8]], [[3qqf|3qqf]], [[3qqg|3qqg]], [[3qqh|3qqh]], [[3qqj|3qqj]], [[3qqk|3qqk]], [[3qql|3qql]], [[3qrt|3qrt]], [[3qru|3qru]], [[3qtq|3qtq]], [[3qtr|3qtr]], [[3qts|3qts]], [[3qtu|3qtu]], [[3qtw|3qtw]], [[3qtx|3qtx]], [[3qtz|3qtz]], [[3qu0|3qu0]], [[3qwj|3qwj]], [[3qwk|3qwk]], [[3qx2|3qx2]], [[3qx4|3qx4]], [[3qxo|3qxo]], [[3qxp|3qxp]], [[3qzf|3qzf]], [[3qzg|3qzg]], [[3qzh|3qzh]], [[3qzi|3qzi]], [[3r1q|3r1q]], [[3r1s|3r1s]], [[3r1y|3r1y]], [[3r28|3r28]], [[3r6x|3r6x]], [[3r71|3r71]], [[3r73|3r73]], [[3r7e|3r7e]], [[3r7i|3r7i]], [[3r7u|3r7u]], [[3r7v|3r7v]], [[3r7y|3r7y]], [[3r83|3r83]], [[3r8l|3r8l]], [[3r8m|3r8m]], [[3r8p|3r8p]], [[3r8u|3r8u]], [[3r8v|3r8v]], [[3r8z|3r8z]], [[3r9d|3r9d]], [[3r9h|3r9h]], [[3r9n|3r9n]], [[3r9o|3r9o]], [[3rah|3rah]], [[3rai|3rai]], [[3rak|3rak]], [[3ral|3ral]], [[3rjc|3rjc]], [[3rk5|3rk5]], [[3rk7|3rk7]], [[3rk9|3rk9]], [[3rkb|3rkb]], [[3rm6|3rm6]], [[3rm7|3rm7]], [[3rmf|3rmf]], [[3rni|3rni]], [[3roy|3roy]], [[3rpo|3rpo]], [[3rpr|3rpr]], [[3rpv|3rpv]], [[3rzb|3rzb]], [[3s00|3s00]], [[3s0o|3s0o]], [[3s1h|3s1h]], [[3sqq|3sqq]]</td></tr> | ||
<tr id='gene'><td class="sblockLbl"><b>[[Gene|Gene:]]</b></td><td class="sblockDat">CDK2 ([http://www.ncbi.nlm.nih.gov/Taxonomy/Browser/wwwtax.cgi?mode=Info&srchmode=5&id=9606 | <tr id='gene'><td class="sblockLbl"><b>[[Gene|Gene:]]</b></td><td class="sblockDat">CDK2 ([http://www.ncbi.nlm.nih.gov/Taxonomy/Browser/wwwtax.cgi?mode=Info&srchmode=5&id=9606 HUMAN])</td></tr> | ||
<tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Cyclin-dependent_kinase Cyclin-dependent kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.11.22 2.7.11.22] </span></td></tr> | <tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Cyclin-dependent_kinase Cyclin-dependent kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.11.22 2.7.11.22] </span></td></tr> | ||
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=3rpy FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=3rpy OCA], [http://www.rcsb.org/pdb/explore.do?structureId=3rpy RCSB], [http://www.ebi.ac.uk/pdbsum/3rpy PDBsum]</span></td></tr> | <tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=3rpy FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=3rpy OCA], [http://pdbe.org/3rpy PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=3rpy RCSB], [http://www.ebi.ac.uk/pdbsum/3rpy PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=3rpy ProSAT]</span></td></tr> | ||
</table> | </table> | ||
== Function == | == Function == | ||
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From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine.<br> | From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine.<br> | ||
</div> | </div> | ||
<div class="pdbe-citations 3rpy" style="background-color:#fffaf0;"></div> | |||
==See Also== | ==See Also== | ||
*[[ | *[[Cyclin-dependent kinase|Cyclin-dependent kinase]] | ||
== References == | == References == | ||
<references/> | <references/> | ||
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</StructureSection> | </StructureSection> | ||
[[Category: Cyclin-dependent kinase]] | [[Category: Cyclin-dependent kinase]] | ||
[[Category: | [[Category: Human]] | ||
[[Category: Alam, R]] | [[Category: Alam, R]] | ||
[[Category: Becker, A]] | [[Category: Becker, A]] |