4lbt: Difference between revisions

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'''Unreleased structure'''
{{STRUCTURE_4lbt|  PDB=4lbt  |  SCENE=  }}
===Endothiapepsin in complex with 100mM acylhydrazone inhibitor===
{{ABSTRACT_PUBMED_24532096}}


The entry 4lbt is ON HOLD  until Paper Publication
==About this Structure==
[[4lbt]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Cryphonectria_parasitica Cryphonectria parasitica]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=4LBT OCA].


Authors: Radeva, N., Heine, A., Winquist, J., Klebe, G.
==Reference==
 
<ref group="xtra">PMID:024532096</ref><references group="xtra"/><references/>
Description: Endothiapepsin in complex with 100mM acylhydrazone inhibitor
[[Category: Cryphonectria parasitica]]
[[Category: Endothiapepsin]]
[[Category: Heine, A.]]
[[Category: Klebe, G.]]
[[Category: Radeva, N.]]
[[Category: Winquist, J.]]
[[Category: Aspartic protease]]
[[Category: Hydrolase]]
[[Category: Hydrolase-hydrolase inhibitor complex]]

Revision as of 12:16, 2 April 2014

Template:STRUCTURE 4lbt

Endothiapepsin in complex with 100mM acylhydrazone inhibitorEndothiapepsin in complex with 100mM acylhydrazone inhibitor

Template:ABSTRACT PUBMED 24532096

About this StructureAbout this Structure

4lbt is a 1 chain structure with sequence from Cryphonectria parasitica. Full crystallographic information is available from OCA.

ReferenceReference

[xtra 1]

  1. Mondal M, Radeva N, Koster H, Park A, Potamitis C, Zervou M, Klebe G, Hirsch AK. Structure-based design of inhibitors of the aspartic protease endothiapepsin by exploiting dynamic combinatorial chemistry. Angew Chem Int Ed Engl. 2014 Mar 17;53(12):3259-63. doi: 10.1002/anie.201309682. , Epub 2014 Feb 14. PMID:24532096 doi:http://dx.doi.org/10.1002/anie.201309682

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OCA