4e47: Difference between revisions

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'''Unreleased structure'''
[[Image:4e47.jpg|left|200px]]


The entry 4e47 is ON HOLD
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{{STRUCTURE_4e47|  PDB=4e47 |  SCENE=  }}


Authors: Walker, J.R., Ouyang, H., Dong, A., Barsyte, D., Vedadi, M., Bountra, C., Weigelt, J., Edwards, A.M., Arrowsmith, C.H., Brown, P.J., Structural Genomics Consortium (SGC)
===SET7/9 in complex with inhibitor (R)-(3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6- sulfonamide and S-adenosylmethionine===


Description: SET7/9 in complex with inhibitor N-(3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl)-1,2,3,4-tetrahtdroisoquinoline-6-sulfonamide and S-adenosylmethionine
 
==About this Structure==
[[4e47]] is a 4 chain structure with sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=4E47 OCA].
[[Category: Histone-lysine N-methyltransferase]]
[[Category: Homo sapiens]]
[[Category: Arrowsmith, C H.]]
[[Category: Barsyte, D.]]
[[Category: Bountra, C.]]
[[Category: Brown, P J.]]
[[Category: Bunnage, M.]]
[[Category: Cook, A.]]
[[Category: Dong, A.]]
[[Category: Edwards, A M.]]
[[Category: Fish, P.]]
[[Category: Ouyang, H.]]
[[Category: Owen, D.]]
[[Category: SGC, Structural Genomics Consortium.]]
[[Category: Tatlock, J.]]
[[Category: Vedadi, M.]]
[[Category: Walker, J R.]]
[[Category: Weigelt, J.]]
[[Category: Chromatin regulator]]
[[Category: Chromosomal protein]]
[[Category: Inhibitor]]
[[Category: Methyltransferase]]
[[Category: Nucleus]]
[[Category: S-adenosylmethionine]]
[[Category: Set domain]]
[[Category: Sgc]]
[[Category: Structural genomics consortium]]
[[Category: Ternary complex]]
[[Category: Transcription]]
[[Category: Transcription regulation]]
[[Category: Transferase]]
[[Category: Transferase-transferase inhibitor complex]]

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