2bpm: Difference between revisions

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|PDB= 2bpm |SIZE=350|CAPTION= <scene name='initialview01'>2bpm</scene>, resolution 2.40&Aring;
|PDB= 2bpm |SIZE=350|CAPTION= <scene name='initialview01'>2bpm</scene>, resolution 2.40&Aring;
|SITE= <scene name='pdbsite=AC1:So4+Binding+Site+For+Chain+D'>AC1</scene>
|SITE= <scene name='pdbsite=AC1:So4+Binding+Site+For+Chain+D'>AC1</scene>
|LIGAND= <scene name='pdbligand=SO4:SULFATE+ION'>SO4</scene> and <scene name='pdbligand=529:(2S)-N-[(3Z)-5-CYCLOPROPYL-3H-PYRAZOL-3-YLIDENE]-2-[4-(2-OXOIMIDAZOLIDIN-1-YL)PHENYL]PROPANAMIDE'>529</scene>
|LIGAND= <scene name='pdbligand=529:(2S)-N-[(3Z)-5-CYCLOPROPYL-3H-PYRAZOL-3-YLIDENE]-2-[4-(2-OXOIMIDAZOLIDIN-1-YL)PHENYL]PROPANAMIDE'>529</scene>, <scene name='pdbligand=SO4:SULFATE+ION'>SO4</scene>
|ACTIVITY= [http://en.wikipedia.org/wiki/Transferred_entry:_2.7.11.1 Transferred entry: 2.7.11.1], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.1.37 2.7.1.37]  
|ACTIVITY= <span class='plainlinks'>[http://en.wikipedia.org/wiki/Non-specific_serine/threonine_protein_kinase Non-specific serine/threonine protein kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.11.1 2.7.11.1] </span>
|GENE=  
|GENE=  
|DOMAIN=
|RELATEDENTRY=
|RESOURCES=<span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=2bpm FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=2bpm OCA], [http://www.ebi.ac.uk/pdbsum/2bpm PDBsum], [http://www.rcsb.org/pdb/explore.do?structureId=2bpm RCSB]</span>
}}
}}


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3-Aminopyrazole inhibitors of CDK2/cyclin A as antitumor agents. 2. Lead optimization., Pevarello P, Brasca MG, Orsini P, Traquandi G, Longo A, Nesi M, Orzi F, Piutti C, Sansonna P, Varasi M, Cameron A, Vulpetti A, Roletto F, Alzani R, Ciomei M, Albanese C, Pastori W, Marsiglio A, Pesenti E, Fiorentini F, Bischoff JR, Mercurio C, J Med Chem. 2005 Apr 21;48(8):2944-56. PMID:[http://www.ncbi.nlm.nih.gov/pubmed/15828833 15828833]
3-Aminopyrazole inhibitors of CDK2/cyclin A as antitumor agents. 2. Lead optimization., Pevarello P, Brasca MG, Orsini P, Traquandi G, Longo A, Nesi M, Orzi F, Piutti C, Sansonna P, Varasi M, Cameron A, Vulpetti A, Roletto F, Alzani R, Ciomei M, Albanese C, Pastori W, Marsiglio A, Pesenti E, Fiorentini F, Bischoff JR, Mercurio C, J Med Chem. 2005 Apr 21;48(8):2944-56. PMID:[http://www.ncbi.nlm.nih.gov/pubmed/15828833 15828833]
[[Category: Homo sapiens]]
[[Category: Homo sapiens]]
[[Category: Non-specific serine/threonine protein kinase]]
[[Category: Protein complex]]
[[Category: Protein complex]]
[[Category: Transferred entry: 2 7.11 1]]
[[Category: Albanese, C.]]
[[Category: Albanese, C.]]
[[Category: Alzani, R.]]
[[Category: Alzani, R.]]
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[[Category: Varasi, M.]]
[[Category: Varasi, M.]]
[[Category: Vulpetti, A.]]
[[Category: Vulpetti, A.]]
[[Category: 529]]
[[Category: SO4]]
[[Category: cell division]]
[[Category: cell division]]
[[Category: cyclin]]
[[Category: cyclin]]
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[[Category: transferase]]
[[Category: transferase]]


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