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==SUBSITE MAPPING OF THE ACTIVE SITE OF HUMAN PANCREATIC ALPHA-AMYLASE USING SUBSTRATES, THE PHARMACOLOGICAL INHIBITOR ACARBOSE, AND AN ACTIVE SITE VARIANT==
==SUBSITE MAPPING OF THE ACTIVE SITE OF HUMAN PANCREATIC ALPHA-AMYLASE USING SUBSTRATES, THE PHARMACOLOGICAL INHIBITOR ACARBOSE, AND AN ACTIVE SITE VARIANT==
<StructureSection load='2cpu' size='340' side='right' caption='[[2cpu]], [[Resolution|resolution]] 2.00&Aring;' scene=''>
<StructureSection load='2cpu' size='340' side='right'caption='[[2cpu]], [[Resolution|resolution]] 2.00&Aring;' scene=''>
== Structural highlights ==
== Structural highlights ==
<table><tr><td colspan='2'>[[2cpu]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Human Human]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=2CPU OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=2CPU FirstGlance]. <br>
<table><tr><td colspan='2'>[[2cpu]] is a 1 chain structure with sequence from [https://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=2CPU OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=2CPU FirstGlance]. <br>
</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=CA:CALCIUM+ION'>CA</scene>, <scene name='pdbligand=CL:CHLORIDE+ION'>CL</scene></td></tr>
</td></tr><tr id='method'><td class="sblockLbl"><b>[[Empirical_models|Method:]]</b></td><td class="sblockDat" id="methodDat">X-ray diffraction, [[Resolution|Resolution]] 2&#8491;</td></tr>
<tr id='NonStdRes'><td class="sblockLbl"><b>[[Non-Standard_Residue|NonStd Res:]]</b></td><td class="sblockDat"><scene name='pdbligand=PCA:PYROGLUTAMIC+ACID'>PCA</scene></td></tr>
<tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=CA:CALCIUM+ION'>CA</scene>, <scene name='pdbligand=CL:CHLORIDE+ION'>CL</scene>, <scene name='pdbligand=PCA:PYROGLUTAMIC+ACID'>PCA</scene></td></tr>
<tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Alpha-amylase Alpha-amylase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=3.2.1.1 3.2.1.1] </span></td></tr>
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=2cpu FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=2cpu OCA], [https://pdbe.org/2cpu PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=2cpu RCSB], [https://www.ebi.ac.uk/pdbsum/2cpu PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=2cpu ProSAT]</span></td></tr>
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=2cpu FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=2cpu OCA], [http://pdbe.org/2cpu PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=2cpu RCSB], [http://www.ebi.ac.uk/pdbsum/2cpu PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=2cpu ProSAT]</span></td></tr>
</table>
</table>
== Function ==
[https://www.uniprot.org/uniprot/AMYP_HUMAN AMYP_HUMAN]
== Evolutionary Conservation ==
== Evolutionary Conservation ==
[[Image:Consurf_key_small.gif|200px|right]]
[[Image:Consurf_key_small.gif|200px|right]]
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__TOC__
__TOC__
</StructureSection>
</StructureSection>
[[Category: Alpha-amylase]]
[[Category: Homo sapiens]]
[[Category: Human]]
[[Category: Large Structures]]
[[Category: Braun, C]]
[[Category: Braun C]]
[[Category: Brayer, G D]]
[[Category: Brayer GD]]
[[Category: Maurus, R]]
[[Category: Maurus R]]
[[Category: Nguyen, N T]]
[[Category: Nguyen NT]]
[[Category: Overall, C M]]
[[Category: Overall CM]]
[[Category: Rydberg, E H]]
[[Category: Rydberg EH]]
[[Category: Sidhu, G]]
[[Category: Sidhu G]]
[[Category: Wang, Y]]
[[Category: Wang Y]]
[[Category: Withers, S G]]
[[Category: Withers SG]]
[[Category: Amylase]]
[[Category: Catalysis]]
[[Category: Diabetes]]
[[Category: Enzyme]]
[[Category: Hydrolase]]
[[Category: Mutagenesis]]
[[Category: Pancreatic]]

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